G-Protein-Coupled Receptors, the largest gene families in the human genome, have become the leading molecular target in 2008.

This year SBS April meeting in Lille, France, followed-up with screening trends report stating that “In 2009, GPCRs are expected to replace protein kinases as the most common molecular target used by HTS laboratories.”

GPCRs are the largest family of cell surface receptors being integral to the number of cellular and physiological functions, including light sensing, smell, appetite control, insulin secretion, and blood pressure modulation.

TimTec GPCR Ligands library, ActiTarg-G, currently counts 2,300 molecules available in various formatting options. ActiTarg-G is the set of molecules that contain chemical lattices present in compounds reported in the technical or patent literature to possess GPCR-ligand properties.

ActiTarg-G is available in various formatting options. Compounds comply with screening purity standards and are in stock for re-supply. Cherry-picking is available.

Contact us may you have any questions or would like to learn more about ActiTarg-G and other TimTec compound library collections, products, and services.